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The semi-synthetic opioid drug hydrocodone is categorized as a Schedule II substance. The Food and Drug Administration (FDA) of the United States has approved this medication for the treatment of pain. The main indication for hydrocodone use is severe chronic pain that cannot be adequately managed with nonopioid alternatives and needs to be treated with opioid analgesia. Because of its antitussive qualities, adults with nonproductive coughs are treated with combination formulations of hydrocodone. In order to produce analgesic effects, hydrocodone activates mu-opioid receptors, acting as an opioid receptor agonist. Hydrocodone also causes the activation of kappa and delta opioid receptors when the drug’s plasma concentration rises above its initial doses. Pain relief with a single ingredient—hydrocodone—is the main focus of this activity.
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